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Virtual Special Issue: Epigenetics 2022.

作者信息

Aldrich Courtney C, Calderón Félix, Conway Stuart J, He Chuan, Hooker Jacob M, Huryn Donna M, Lindsley Craig W, Liotta Dennis C, Müller Christa E

出版信息

ACS Pharmacol Transl Sci. 2022 Sep 9;5(10):829-834. doi: 10.1021/acsptsci.2c00169. eCollection 2022 Oct 14.

Abstract
摘要

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本文引用的文献

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Small-Molecule Inhibitors of the MLL1 CXXC Domain, an Epigenetic Reader of DNA Methylation.
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Conformational-Design-Driven Discovery of EZM0414: A Selective, Potent SETD2 Inhibitor for Clinical Studies.
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